| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Beta-arrestin-1 |
|---|
| Ligand | BDBM224017 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | beta-Arrestin Assay |
|---|
| EC50 | 310±n/a nM |
|---|
| Citation |  Tounge, BA; Bayoumy, S; Kuo, LC; Dax, SL Substituted 3-dialkylaminomethyl-piperidin-4-yl-benzamides and methods of making and using same US Patent US10836728 Publication Date 11/17/2020 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Beta-arrestin-1 |
|---|
| Name: | Beta-arrestin-1 |
|---|
| Synonyms: | ARR1 | ARRB1 | ARRB1_HUMAN | Arrestin, beta 1 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 47062.57 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_13177715 |
|---|
| Residue: | 418 |
|---|
| Sequence: | MGDKGTRVFKKASPNGKLTVYLGKRDFVDHIDLVDPVDGVVLVDPEYLKERRVYVTLTCA
FRYGREDLDVLGLTFRKDLFVANVQSFPPAPEDKKPLTRLQERLIKKLGEHAYPFTFEIP
PNLPCSVTLQPGPEDTGKACGVDYEVKAFCAENLEEKIHKRNSVRLVIRKVQYAPERPGP
QPTAETTRQFLMSDKPLHLEASLDKEIYYHGEPISVNVHVTNNTNKTVKKIKISVRQYAD
ICLFNTAQYKCPVAMEEADDTVAPSSTFCKVYTLTPFLANNREKRGLALDGKLKHEDTNL
ASSTLLREGANREILGIIVSYKVKVKLVVSRGGLLGDLASSDVAVELPFTLMHPKPKEEP
PHREVPENETPVDTNLIELDTNDDDIVFEDFARQRLKGMKDDKEEEEDGTGSPQLNNR
|
|
|
|---|
| BDBM224017 |
|---|
| n/a |
|---|
| Name | BDBM224017 |
|---|
| Synonyms: | (+)-Morphine | US10752592, Compound morphine | US10836728, Compound Morphine | US11534436, Compound morphine |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C17H19NO3 |
|---|
| Mol. Mass. | 285.3377 |
|---|
| SMILES | CN1CC[C@]23[C@@H]4Oc5c2c(C[C@H]1[C@H]3C=C[C@H]4O)ccc5O |c:16| |
|---|
| Structure | 
|
|---|
Search and Browse
