| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Bromodomain-containing protein 4 [44-167] |
|---|
| Ligand | BDBM483491 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | Alpha-assay |
|---|
| IC50 | 24.3±n/a nM |
|---|
| Citation |  Landau, SB; Kagey, MH Treatment of conditions associated with hyperinsulinaemia US Patent US10925881 Publication Date 2/23/2021 |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Bromodomain-containing protein 4 [44-167] |
|---|
| Name: | Bromodomain-containing protein 4 [44-167] |
|---|
| Synonyms: | BRD4 | BRD4 bromodomain 1 | BRD4_HUMAN | Brd4-1 | HUNK1 |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 14738.39 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | O60885[44-167] |
|---|
| Residue: | 124 |
|---|
| Sequence: | NPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKT
PMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINE
LPTE
|
|
|
|---|
| BDBM483491 |
|---|
| n/a |
|---|
| Name | BDBM483491 |
|---|
| Synonyms: | US10925881, Name (S)-JQ35 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C27H34ClN7OS |
|---|
| Mol. Mass. | 540.123 |
|---|
| SMILES | CN1CCN(CCCNC(=O)C[C@@H]2N=C(c3c(C)c(C)sc3-n3c(C)nnc23)c2ccc(Cl)cc2)CC1 |r,c:13| |
|---|
| Structure | 
|
|---|
Search and Browse
