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Assay Method Information

Assay Name:  ChEMBL_978570 (CHEMBL2421940)
Description:  Antagonist activity at CB2 receptor in HEK293 cells assessed as increase in CP-55,940 EC50 measuring inhibition of forskolin-stimulated cAMP accumulation at 1 uM incubated 20 mins prior to CP-55,940 addition measured after 7 mins by spectrophotometry (Rvb = 4.21+/-1.16 nM)
Affinity data for this assay
 

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Last update November 1, 2007
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