Assay Method Information |
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| ChEMBL_1901767 (CHEMBL4403989) |
Description: | Inhibition of PI3Kgamma in mouse RAW264 cells assessed as reduction in C5a anaphylatoxin trifluoroacetate salt-induced AKT phosphorylation at T208 residue preincubated for 1 hr followed by C5a anaphylatoxin trifluoroacetate salt addition and measured after 3 mins by QuantaBlu substrate based fluorescence assay |
Affinity data for this assay | |
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