Assay Method Information |
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| ChEMBL_1878653 (CHEMBL4380047) |
Description: | Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as inhibition of rosiglitazone-induced N-terminal biotinylated co-activator SRC1 box2 peptide recruitment measured after 30 mins by TR-FRET assay |
Affinity data for this assay | |
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