Assay Method Information |
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| ChEMBL_2132578 (CHEMBL4842093) |
Description: | Partial agonist activity at D2 receptor (unknown origin) expressed in HEK293T cells co-expressing Rluc8-tagged Galpahi1 assessed as Galphai1 dissociation preincubated for 2 mins with coelenterazine followed by compound addition and measured after 2 mins by BRET assay |
Affinity data for this assay | |
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