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Assay Method Information

Assay Name:  ChEMBL_1437089 (CHEMBL3381103)
Description:  Modulation of BCRP1 mediated drug efflux in mitoxantrone-resistant human MES-SA cells assessed as accumulation of hoechst 33342 incubated for 15 mins prior to rhodamine-123 addition measured after 90 mins by fluorescence analysis
Affinity data for this assay
 

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Last update November 1, 2007
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