Assay Method Information |
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| Coactivator Peptide Competitive FP Assay (IC50/EC50) |
Description: | AR functionality was determined by fluorescence polarization (excitation @485 nm, emission @ 530 nm) assay, which measures fluorescently labeled SRC2-3 peptide displacement from DHT-bound AR-LBD. |
Affinity data for this assay | |
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