Assay Method Information |
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| ChEMBL_1766898 (CHEMBL4202145) |
Description: | Inhibition of human VMAT2 expressed in HEK293 cell membranes assessed as reduction in [3H[-5HT uptake pre-incubated for 10 mins before [3H[-5HT addition and measured after 6 mins |
Affinity data for this assay | |
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