Assay Method Information |
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| ChEMBL_1766053 (CHEMBL4201300) |
Description: | Antagonist activity at UT receptor in Sprague-Dawley rat thoracic aortic ring assessed as reduction in urotensin-2-induced contraction by measuring pEC50 for human urotensin-2-induced contraction at 1 uM pre-incubated for 30 mins before urotensin-2 stimulation (Rvb = 8.59 +/- 0.12 No_unit) |
Affinity data for this assay | |
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