Compile Data Set for Download or QSAR
Found 31 of affinity data for UniProtKB/TrEMBL: Q8VIJ5
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50531967(Pugnac)copy SMILEScopy InChI
Affinity DataKi:  50nMAssay Description:Inhibition of rat spleen OGAMore data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50041556(CHEMBL3358418)copy SMILEScopy InChI
Affinity DataEC50: <200nMAssay Description:Inhibition of OGA in rat B35 cells after 16 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SK0PubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50041557(CHEMBL3358419)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of OGA in rat B35 cells after 16 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SK0PubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50323697((3AR,5R,6S,7R,7AR)-2-(ETHYLAMINO)-5-(HYDROXYMETHYL...)copy SMILEScopy InChI
Affinity DataEC50:  30nMAssay Description:Inhibition of O-GlcNAcase in rat PC12 cells assessed as induction of OGlcNAcylation after 24 hrs by Western blot methodMore data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513930(CHEMBL4543991)copy SMILEScopy InChI
Affinity DataEC50:  176nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513931(CHEMBL4444446)copy SMILEScopy InChI
Affinity DataEC50:  11nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513934(CHEMBL4443587)copy SMILEScopy InChI
Affinity DataEC50:  1.70nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50323697((3AR,5R,6S,7R,7AR)-2-(ETHYLAMINO)-5-(HYDROXYMETHYL...)copy SMILEScopy InChI
Affinity DataEC50:  14nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513955(CHEMBL4483089)copy SMILEScopy InChI
Affinity DataEC50:  37nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513956(CHEMBL4448352)copy SMILEScopy InChI
Affinity DataEC50:  443nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513957(CHEMBL4456515)copy SMILEScopy InChI
Affinity DataEC50:  509nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM141965(US8927507, 16)copy SMILEScopy InChI
Affinity DataEC50:  152nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513958(CHEMBL4473252)copy SMILEScopy InChI
Affinity DataEC50:  177nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513951(CHEMBL4583010)copy SMILEScopy InChI
Affinity DataEC50:  445nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513950(CHEMBL4454814)copy SMILEScopy InChI
Affinity DataEC50:  224nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM205421(US9243020, 4 | US9815861, Example 4)copy SMILEScopy InChI
Affinity DataEC50:  358nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513939(CHEMBL4516713)copy SMILEScopy InChI
Affinity DataEC50:  33nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM142083(US8933040, 7)copy SMILEScopy InChI
Affinity DataEC50:  165nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513947(CHEMBL4545886)copy SMILEScopy InChI
Affinity DataEC50:  28nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513960(CHEMBL4561925)copy SMILEScopy InChI
Affinity DataEC50:  41nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM205425(US9243020, 20 | US9815861, Example 20)copy SMILEScopy InChI
Affinity DataEC50:  31nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM205428(US9243020, 33 | US9815861, Example 33)copy SMILEScopy InChI
Affinity DataEC50:  58nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM205423(US9243020, 17 | US9815861, Example 17)copy SMILEScopy InChI
Affinity DataEC50:  34nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM205424(US9243020, 19 | US9815861, Example 19)copy SMILEScopy InChI
Affinity DataEC50:  53nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM205422(US9243020, 9 | US9815861, Example 9)copy SMILEScopy InChI
Affinity DataEC50:  307nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513949(CHEMBL4476839)copy SMILEScopy InChI
Affinity DataEC50:  328nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513933(CHEMBL4513613)copy SMILEScopy InChI
Affinity DataEC50:  2.40E+3nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM205420(US9243020, 2 | US9815861, Example 2)copy SMILEScopy InChI
Affinity DataEC50:  364nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50513940(CHEMBL4586062)copy SMILEScopy InChI
Affinity DataEC50:  119nMAssay Description:Inhibition of OGA in rat PC12 cells assessed as OGlcNAcylated protein level incubated for 24 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0QMHPubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50041554(CHEMBL3358417)copy SMILEScopy InChI
Affinity DataEC50:  200nMAssay Description:Inhibition of OGA in rat B35 cells after 16 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SK0PubMed
TargetProtein O-GlcNAcase(Rattus norvegicus)
Nankai University

Curated by ChEMBL
LigandPNGBDBM50041555(CHEMBL1379586)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of OGA in rat B35 cells after 16 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4SK0PubMed