42 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
PMID
Data
Article Title
Organization
Synthetic, enzyme kinetic, and protein crystallographic studies of C-ß-d-glucopyranosyl pyrroles and imidazoles reveal and explain low nanomolar inhibition of human liver glycogen phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Thessaly
Synthesis of (benzimidazol-2-yl)aniline derivatives as glycogen phosphorylase inhibitors.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
Egypt National Research Centre
2-Oxo-1,2-dihydropyridinyl-3-yl amide-based GPa inhibitors: Design, synthesis and structure-activity relationship study.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
Griffith University
4(5)-Aryl-2-C-glucopyranosyl-imidazoles as New Nanomolar Glucose Analogue Inhibitors of Glycogen Phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Glucose-derived spiro-isoxazolines are anti-hyperglycemic agents against type 2 diabetes through glycogen phosphorylase inhibition.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
Universit£
Structure based inhibitor design targeting glycogen phosphorylase B. Virtual screening, synthesis, biochemical and biological assessment of novel N-acyl-ß-d-glucopyranosylamines.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Thessaly
New synthesis of 3-(ß-D-glucopyranosyl)-5-substituted-1,2,4-triazoles, nanomolar inhibitors of glycogen phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Synthesis, enzyme kinetics and computational evaluation of N-(ß-D-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
C-Glucopyranosyl-1,2,4-triazoles As New Potent Inhibitors of Glycogen Phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Synthesis of tartaric acid analogues of FR258900 and their evaluation as glycogen phosphorylase inhibitors.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
The binding of C5-alkynyl and alkylfurano[2,3-d]pyrimidine glucopyranonucleosides to glycogen phosphorylase b: synthesis, biochemical and biological assessment.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Thessaly
Binding evaluation of fragment-based scaffolds for probing allosteric enzymes.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
Universit£
1-(3-Deoxy-3-fluoro-beta-d-glucopyranosyl) pyrimidine derivatives as inhibitors of glycogen phosphorylase b: Kinetic, crystallographic and modelling studies.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
National Hellenic Research Foundation
Terpenoids. III: Synthesis and biological evaluation of 23-hydroxybetulinic acid derivatives as novel inhibitors of glycogen phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
China Pharmaceutical University
Practical synthesis of bredemolic acid, a natural inhibitor of glycogen phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
China Pharmaceutical University
Pentacyclic triterpenes. Part 3: Synthesis and biological evaluation of oleanolic acid derivatives as novel inhibitors of glycogen phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
China Pharmaceutical University
N-(4-Substituted-benzoyl)-N'-(ß-d-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methods.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Design and synthesis of novel photoaffinity probes for study of the target proteins of oleanolic acid.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
China Pharmaceutical University
Halogen-substituted (C-ß-D-glucopyranosyl)-hydroquinone regioisomers: synthesis, enzymatic evaluation and their binding to glycogen phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
National Hellenic Research Foundation
Ligand-based modelling followed by synthetic exploration unveil novel glycogen phosphorylase inhibitory leads.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
Applied Science University
Identification of pentacyclic triterpenes derivatives as potent inhibitors against glycogen phosphorylase based on 3D-QSAR studies.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
Chinese Academy of Sciences
Efficient synthesis and biological evaluation of epiceanothic acid and related compounds.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
China Pharmaceutical University
The binding ofß-d-glucopyranosyl-thiosemicarbazone derivatives to glycogen phosphorylase: A new class of inhibitors.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
National Hellenic Research Foundation
Synthesis of 3-deoxypentacyclic triterpene derivatives as inhibitors of glycogen phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
China Pharmaceutical University
Synthesis of 1-(D-glucopyranosyl)-1,2,3-triazoles and their evaluation as glycogen phosphorylase inhibitors.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Synthesis and glycogen phosphorylase inhibitory activity of N-(beta-D-glucopyranosyl)amides possessing 1,4-benzodioxane moiety.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Synthesis and structure-activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Glucose-based spiro-heterocycles as potent inhibitors of glycogen phosphorylase.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Fructose-1,6-bisphosphatase inhibitors. 1. Purine phosphonic acids as novel AMP mimics.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
Metabasis Therapeutics
Novel design principle validated: glucopyranosylidene-spiro-oxathiazole as new nanomolar inhibitor of glycogen phosphorylase, potential antidiabetic agent.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Evaluation of novel hyphodermin derivatives as glycogen phosphorylase a inhibitors.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
Griffith University
Iminosugars as potential inhibitors of glycogenolysis: structural insights into the molecular basis of glycogen phosphorylase inhibition.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
The National Hellenic Research Foundation
Pentacyclic triterpenes. Part 2: Synthesis and biological evaluation of maslinic acid derivatives as glycogen phosphorylase inhibitors.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
China Pharmaceutical University
Synthesis, screening and docking of small heterocycles as glycogen phosphorylase inhibitors.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
Griffith University
Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methods.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
A multidisciplinary study of 3-(?-d-glucopyranosyl)-5-substituted-1,2,4-triazole derivatives as glycogen phosphorylase inhibitors: Computation, synthesis, crystallography and kinetics reveal new potent inhibitors.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Nanomolar Inhibitors of Glycogen Phosphorylase Based on?-d-Glucosaminyl Heterocycles: A Combined Synthetic, Enzyme Kinetic, and Protein Crystallography Study.![EBI](/images/logo_chembl.png)
![EBI](/images/logo_chembl.png)
University of Debrecen
Identification of inhibitors that target dual-specificity phosphatase 5 provide new insights into the binding requirements for the two phosphate pockets.![BDB](/images/logo_bindingdb.png)
![BDB](/images/logo_bindingdb.png)
Texas Wesleyan University
Extended radioligand binding profile of iloperidone: a broad spectrum dopamine/serotonin/norepinephrine receptor antagonist for the management of psychotic disorders.![BDB](/images/logo_bindingdb.png)
![BDB](/images/logo_bindingdb.png)
Novartis Pharma
Synthesis and urease enzyme inhibitory effects of some dicoumarols.![BDB](/images/logo_bindingdb.png)
![BDB](/images/logo_bindingdb.png)
University of Karachi