null
SMILES CC(C)OC(=O)c1cn(Cc2c(F)cccc2F)c2sc(c(CN(C)Cc3ccccc3)c2c1=O)-c1ccc(NC(=O)C(C)C)cc1
InChI Key InChIKey=RANJJVIMTOIWIN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50067485
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Chemical Industries, Ltd.
Curated by ChEMBL
Takeda Chemical Industries, Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:The Compound was tested for the concentration to inhibit 50% of [125 I ]leuprorelin binding to the cloned human Leutinizing releasing hormone recepto...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Takeda Chemical Industries, Ltd.
Curated by ChEMBL
Takeda Chemical Industries, Ltd.
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:The compound was tested for the concentration to inhibit 50% of [125 I]leuprorelin binding to Leutinizing releasing hormone receptor in the membrane ...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Takeda Chemical Industries, Ltd.
Curated by ChEMBL
Takeda Chemical Industries, Ltd.
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:The compound was tested for the concentration to inhibit 50% of [125 I]leuprorelin binding to Leutinizing releasing hormone receptor the membrane fra...More data for this Ligand-Target Pair