null
SMILES CC(C)(C)OC(=O)N1CCN(CC1)S(=O)(=O)c1ccc(NC(=O)C=C)cc1F
InChI Key InChIKey=ANNVTFXGUOTPFJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50420457
Affinity DataIC50: 51nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase K(Homo sapiens (Human))
Evotec (UK) Ltd.
Curated by ChEMBL
Evotec (UK) Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human recombinant TG1 by fluorescent transamidation assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Evotec (UK) Ltd.
Curated by ChEMBL
Evotec (UK) Ltd.
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human recombinant TG2 by fluorescent transamidation assayMore data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase E(Homo sapiens (Human))
Evotec (UK) Ltd.
Curated by ChEMBL
Evotec (UK) Ltd.
Curated by ChEMBL
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of thrombin activated human TG3 by fluorescent transamidation assayMore data for this Ligand-Target Pair