null
SMILES O=c1cc(oc2ccccc12)-c1ccccc1
InChI Key InChIKey=VHBFFQKBGNRLFZ-UHFFFAOYSA-N
PDB links: 2 PDB IDs match this monomer.
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50028962
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
University of Oulu
Curated by ChEMBL
University of Oulu
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of human 6XHis-tagged TNKS1 SAM-ART domain (1030 to 1317 amino acid residues) by fluorescence assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
University of Oulu
Curated by ChEMBL
University of Oulu
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of human 6XHis-tagged TNKS2 ART domain (946 to 1161 amino acid residues) expressed in Escherichia coli Rosetta2 (DE3) by fluorescence assa...More data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human recombinant ARTD1 by fluorescence assayMore data for this Ligand-Target Pair