null
SMILES FC(F)Cn1c2cc(ccc2oc1=O)-c1ccc(C[C@H](NC(=O)[C@@H]2CNCCCO2)C#N)cc1
InChI Key InChIKey=ANPJTTUBCRFBKA-RXVVDRJESA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50195248
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
Curated by ChEMBL
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of DPP1 in human U937 cells using Gly-Phe-AFC as substrate preincubated for 60 mins followed by substrate addition by fluorescence assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
Curated by ChEMBL
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
Curated by ChEMBL
CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human recombinant DPP1 using Gly-Arg-AMC as substrate preincubated for 30 mins followed by substrate addition by fluorometric assayMore data for this Ligand-Target Pair