null
SMILES Cc1sc-2c(c1C)C(=NC(CC(=O)NCCN1CCOCC1)c1nnc(C)n-21)c1ccc(Cl)cc1
InChI Key InChIKey=KULOTNHGHJGDQB-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 223494
TargetBromodomain-containing protein 4 [368-440](Homo sapiens (Human))
Dana-Farber Cancer Institute, Inc.
US Patent
Dana-Farber Cancer Institute, Inc.
US Patent
Affinity DataIC50: 29.5nMAssay Description:All reagents were diluted in 50 mM HEPES, 100 mM NaCl, 0.1% BSA, pH 7.4 supplemented with 0.05% CHAPS and allowed to equilibrate to room temperature ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4 [75-147](Homo sapiens (Human))
Dana-Farber Cancer Institute, Inc.
US Patent
Dana-Farber Cancer Institute, Inc.
US Patent
Affinity DataIC50: 85nMAssay Description:All reagents were diluted in 50 mM HEPES, 100 mM NaCl, 0.1% BSA, pH 7.4 supplemented with 0.05% CHAPS and allowed to equilibrate to room temperature ...More data for this Ligand-Target Pair