null
SMILES CNc1ccc(Oc2sc(C(N)=O)c3CCc4cnsc4-c23)cn1
InChI Key InChIKey=LFUBEMFSRYUGLW-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50248645
TargetCyclin-dependent kinase 8(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd.
Curated by ChEMBL
Takeda Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataEC50: 0.580nMAssay Description:Inhibition of CDK8 in human SW620 cells assessed as decrease in STAT1 phosphorylation at Ser727 after 2 hrs by Western blot methodMore data for this Ligand-Target Pair