null
SMILES CCC(=O)N1CCc2ccc(cc2CC1)C(=O)CCCN1CCC(CC1)c1ccc(Cl)cc1
InChI Key InChIKey=NZHJHYYMLWBZAI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50357502
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd
Curated by ChEMBL
Takeda Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Displacement of [125I]-MCH(4-19) from human MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Takeda Pharmaceutical Co., Ltd
Curated by ChEMBL
Takeda Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO cells assessed as inhibition of MCH-stimulated arachidonic acid releaseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Displacement of [125I]-MCH(4-19) from rat MCHR1 expressed in CHO cellsMore data for this Ligand-Target Pair