null
SMILES C[C@H]([C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H]1CCCN1C(=O)[C@@H](N)Cc1ccc(O)cc1)C(N)=O)c1ccccc1
InChI Key InChIKey=XEDWKSFZTLIHLE-VRTFYRIBSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50139015
Affinity DataKi: 0.800nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Displacement of [3H]-endomorphin-2 from Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.67nMAssay Description:Displacement of [3H]-DAMGO from Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(MOUSE)
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 9.15nMAssay Description:Inhibition of Mu opioid receptor of mouse vas deferensMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(GUINEA PIG)
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Biological Research Center of the Hungarian Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 3.46nMAssay Description:Inhibition of Opioid receptor mu 1 of guinea pig ileumMore data for this Ligand-Target Pair