null
SMILES Cn1ncnc1[C@H]1[C@@H](Nc2cc(F)cc3c2c1n[nH]c3=O)c1ccc(F)cc1
InChI Key InChIKey=HWGQMRYQVZSGDQ-HOTGVXAUSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50145156
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Health& Science University
Curated by ChEMBL
Health& Science University
Curated by ChEMBL
Affinity DataIC50: 322nMAssay Description:Inhibition of recombinant human TNKS1 ADP-ribosyltransferase/sterile alpha motif domain expressed in Escherichia coli BL21(DE3) preincubated for 15 m...More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Health& Science University
Curated by ChEMBL
Health& Science University
Curated by ChEMBL
Affinity DataIC50: 324nMAssay Description:Inhibition of recombinant human TNKS1 ADP-ribosyltransferase/sterile alpha motif domain expressed in Escherichia coli BL21(DE3) preincubated for 15 m...More data for this Ligand-Target Pair