null

SMILES C[C@@H]1CCc2c(Br)c(F)c(Br)cc2N1C=O

InChI Key InChIKey=ZZLQPWXVZCPUGC-ZCFIWIBFSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50280395   

TargetRap guanine nucleotide exchange factor 4(Homo sapiens (Human))
Institute for Research in Cancer and Allied Diseases

Curated by ChEMBL
LigandPNGBDBM50280395(CHEMBL4171480)copy SMILEScopy InChI
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPAC2 expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine nucleotide exchange ac...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C4Z83PubMed
TargetRap guanine nucleotide exchange factor 4(Homo sapiens (Human))
Institute for Research in Cancer and Allied Diseases

Curated by ChEMBL
LigandPNGBDBM50280395(CHEMBL4171480)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Antagonist activity at recombinant full length EPAC2 (unknown origin) assessed as inhibition of cAMP-mediated Rap1b-BODIPY GDP nucleotide exchange ac...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TB19FFPubMed