null
SMILES FC(F)(F)c1cccc(c1)-c1ccc(Oc2ccc(cc2C#N)S(=O)(=O)Nc2ncns2)c(c1)-c1ccnc(CNCCC2CCNCC2)c1
InChI Key InChIKey=WSPHMGORSRQULF-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50451447
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
SiteOne Therapeutics
Curated by ChEMBL
SiteOne Therapeutics
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human Nav1.5 expressed in HEK293 cells by electrophysiology assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
SiteOne Therapeutics
Curated by ChEMBL
SiteOne Therapeutics
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human Nav1.5 expressed in HEK cells by automated patchXpress electrophysiology methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
SiteOne Therapeutics
Curated by ChEMBL
SiteOne Therapeutics
Curated by ChEMBL
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition of human Nav1.5 by Q-patch clamp electrophysiology methodMore data for this Ligand-Target Pair