null
SMILES COc1ncc(cn1)-c1nc(C(=O)NC(N)=N)c(N)nc1N
InChI Key InChIKey=XFGYFQDKMRBURI-UHFFFAOYSA-N
PDB links: 1 PDB ID matches this monomer.
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50529264
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Wollongong
Curated by ChEMBL
University of Wollongong
Curated by ChEMBL
Affinity DataKi: 204nMAssay Description:Inhibition of human kidney uPA using fluorogenic Z-Pyr-Gly-Arg-MCA as substrate measured after 15 mins by fluorometric analysisMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University of Wollongong
Curated by ChEMBL
University of Wollongong
Curated by ChEMBL
Affinity DataKi: 204nMAssay Description:Inhibition of human uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair
Affinity DataKi: 956nMAssay Description:Inhibition of mouse uPA using Z-Gly-Gly-Arg-AMC as substrate measured for 15 mins by fluorometric assayMore data for this Ligand-Target Pair