null
SMILES COc1ccc2nnn(CC(=O)N[C@@H](C)c3ccc(C)cc3)c(=O)c2c1
InChI Key InChIKey=MPFIBOVPLHCEFO-ZDUSSCGKSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 263453
TargetProbable G-protein coupled receptor 139(Homo sapiens (Human))
Takeda Pharmaceutical Company Limited
US Patent
Takeda Pharmaceutical Company Limited
US Patent
Affinity DataEC50: 10nMAssay Description:Agonist activity at human GPR139 expressed in CHO-TRex cells assessed as stimulation of calcium signalling incubated for 15 mins by FLIPR assayMore data for this Ligand-Target Pair