null
SMILES Cc1ccn(n1)-c1ccc(C(=O)N2Cc3cccn3Cc3ccccc23)c(Cl)c1
InChI Key InChIKey=JXKQHDZUZGKDGO-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50177593
TargetVasopressin V2 receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
Affinity DataEC50: 0.700nMAssay Description:Agonist activity at V2 receptor (unknown origin) by cAMP accumulation assayMore data for this Ligand-Target Pair
TargetVasopressin V1a receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
Affinity DataEC50: 465nMAssay Description:Activity at human vasopressin V1a receptor expressed in CHO cells by NFAT-luciferase gene reporter assayMore data for this Ligand-Target Pair
Affinity DataEC50: 125nMAssay Description:Activity at human oxytocin receptor expressed in CHO cells by NFAT-luciferase gene reporter assayMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
Affinity DataEC50: 39.9nMAssay Description:Activity at human vasopressin V2 receptor expressed in CHO cells by NFAT-luciferase gene reporter assayMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
UMR7200 CNRS/Universit£ de Strasbourg
Curated by ChEMBL
Affinity DataEC50: 0.740nMAssay Description:Binding to human V2 receptor expressed in LV2 cells by cAMP productionMore data for this Ligand-Target Pair