null
SMILES CC(=O)N1CCc2c(C1)c(nn2C1CCNCC1)N1CCCc2cc(-c3cnn(C)c3)c(cc12)C(F)F
InChI Key InChIKey=LHZXBZYVTILAIU-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50269907
TargetCREB-binding protein(Homo sapiens (Human))
Genentech, Inc. , 1 DNA Way, South San Francisco, California 94080, United States.
Curated by ChEMBL
Genentech, Inc. , 1 DNA Way, South San Francisco, California 94080, United States.
Curated by ChEMBL
Affinity DataIC50: 690nMAssay Description:Inhibition of Halo-tagged histone H3.3 binding to NanoLuc luciferase conjugated human CBP expressed in HEK293 cells after overnight incubation by BRE...More data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Genentech, Inc. , 1 DNA Way, South San Francisco, California 94080, United States.
Curated by ChEMBL
Genentech, Inc. , 1 DNA Way, South San Francisco, California 94080, United States.
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Displacement of biotinylated histone H3K14 peptide ligand from human recombinant His-tagged CBP measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Genentech, Inc. , 1 DNA Way, South San Francisco, California 94080, United States.
Curated by ChEMBL
Genentech, Inc. , 1 DNA Way, South San Francisco, California 94080, United States.
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Displacement of biotinylated histone H3K14 peptide ligand from human recombinant His-tagged BRD4 bromodomain-1 measured after 10 mins by TR-FRET assa...More data for this Ligand-Target Pair