null
SMILES CC1(CCN(CCc2cnn(c2)-c2nccc3c2nc[nH]c3=O)CC1)c1cccc(Cl)c1
InChI Key InChIKey=BPCMQRINPLMHHT-UHFFFAOYSA-N
PDB links: 1 PDB ID matches this monomer.
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50513360
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research
Curated by ChEMBL
Institute of Cancer Research
Curated by ChEMBL
Affinity DataIC50: 107nMAssay Description:Inhibition of N-terminal His-tagged recombinant human KDM4A (1 to 359 residues) expressed in Escherichia coli assessed as decrease in demethylation o...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Institute of Cancer Research
Curated by ChEMBL
Institute of Cancer Research
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of KDM5B (unknown origin) assessed as decrease in demethylation of substrate using peptide (H3(1-21)K4-Me3-GGKBiotin) as substrate and 2OG...More data for this Ligand-Target Pair
TargetLysine-specific demethylase 4B(Homo sapiens (Human))
Institute of Cancer Research
Curated by ChEMBL
Institute of Cancer Research
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human KDM4B (1 to 500 residues) expressed in baculovirus infected Sf9 insect cells assessed as decrea...More data for this Ligand-Target Pair