null
SMILES Fc1ccc(cc1Cl)C(=O)N1CCC(F)(CNCCOc2ccccc2)CC1
InChI Key InChIKey=DXWRIDGYFFSIIY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 9 hits for monomerid = 433474
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
NEUROLIXIS; UNIVERSITE JAGELLONE
US Patent
NEUROLIXIS; UNIVERSITE JAGELLONE
US Patent
Affinity DataKi: 0.0610nMAssay Description:5-HT1A: Radioligand binding was performed using membranes from CHO-K1 cells stably transfected with the human 5-HT1A receptor. All assays were carrie...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
NEUROLIXIS; UNIVERSITE JAGELLONE
US Patent
NEUROLIXIS; UNIVERSITE JAGELLONE
US Patent
Affinity DataKi: 0.0617nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor stably expressed in CHO-K1 cell membranes measured after 60 mins by Microbeta2 scintillation...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
NEUROLIXIS; UNIVERSITE JAGELLONE
US Patent
NEUROLIXIS; UNIVERSITE JAGELLONE
US Patent
Affinity DataKi: 0.0617nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5HT1A receptor stably expressed in CHO-K1 cell membranes measured after 60 mins by microbeta2 sc...More data for this Ligand-Target Pair
Affinity DataKi: 380nMAssay Description:Alpha1-adrenergic Receptor: Radioligand binding was performed using tissue (rat cortex). All assays were carried out in duplicates. 50 μL workin...More data for this Ligand-Target Pair
Affinity DataKi: 513nMAssay Description:Displacement of [3H]-prazosin from alpha1 adrenergic receptor in rat cortex measured after 30 mins by microbeta2 scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 513nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenergic receptor in rat cortex membranes measured after 30 mins by Microbeta2 scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]-methylspiperone from recombinant human D2 receptor stably expressed in CHO-K1 cell membranes measured after 60 mins by microbeta...More data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]methylspiperone from human D2 receptor stably expressed in CHO-K1 cell membranes measured after 60 mins by Microbeta2 scintillati...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:D2 Dopamine Receptor:Radioligand binding was performed using membranes from CHO-K1 cells stably transfected with the human D2 receptor. All assays we...More data for this Ligand-Target Pair