null
SMILES O=C(C1CC1)c1ccc(OCCCc2c[nH]cn2)cc1
InChI Key InChIKey=ACQBHJXEAYTHCY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50458225
TargetHistamine H3 receptor(Homo sapiens (Human))
CSIR-Central Drug Research Institute
Curated by ChEMBL
CSIR-Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human H3R expressed in HEK293 cell membranes incubated for 90 mins by liquid scintillation counting...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
CSIR-Central Drug Research Institute
Curated by ChEMBL
CSIR-Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Binding affinity to human H3RMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
CSIR-Central Drug Research Institute
Curated by ChEMBL
CSIR-Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Inhibition of human histamine H3 receptorMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
CSIR-Central Drug Research Institute
Curated by ChEMBL
CSIR-Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]UR-PI294 from human SP-FLAG-tagged H3R expressed in HEK293T cells measured after 60 to 120 mins by liquid scintillation counting ...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
CSIR-Central Drug Research Institute
Curated by ChEMBL
CSIR-Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 63nMAssay Description:Binding affinity to human H3RMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
CSIR-Central Drug Research Institute
Curated by ChEMBL
CSIR-Central Drug Research Institute
Curated by ChEMBL
Affinity DataKi: 224nMAssay Description:Displacement of [3H] N-alpha methylhistamine from human recombinant histamine H3 receptor expressed in HEK293 cells measured after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB-603 from human recombinant adenosine A2B receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]PSB-11 from human recombinant adenosine A3 receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair