null
SMILES CC(C)(C)c1ccc(cc1)C(=O)Nc1cn2cc(ccc2n1)-n1ccnc1
InChI Key InChIKey=SMJAMOAYGIVKRI-UHFFFAOYSA-N
PDB links: 1 PDB ID matches this monomer.
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50334268
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
PharmaDesign, Inc.
Curated by ChEMBL
PharmaDesign, Inc.
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of ASK1 assessed as phosphorylated fluorescent peptide by mobility shift assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
PharmaDesign, Inc.
Curated by ChEMBL
PharmaDesign, Inc.
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Competitive inhibition of human recombinant N-terminal FLAG-tagged ASK1 expressed in baculovirus infected Sf2 cells after 60 mins by scintillation co...More data for this Ligand-Target Pair