null
SMILES O=C(Cc1ccccc1)Nc1nnc(CCCCCc2nnc(NC(=O)Cc3ccccc3)s2)s1
InChI Key InChIKey=IAGMXTIWZLWUOZ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 108454
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Calithera Biosciences Inc.
US Patent
Calithera Biosciences Inc.
US Patent
Affinity DataIC50: 1.40E+3nMAssay Description:Compounds were assessed for their ability to inhibit the enzymatic activity of a recombinant form of Glutaminase 1 (GAC) using a biochemical assay th...More data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Calithera Biosciences Inc.
US Patent
Calithera Biosciences Inc.
US Patent
Affinity DataIC50: 380nMAssay Description:Inhibition of recombinant 6His-tagged GLS1 KGA isoform (unknown origin) (63 to 669 residues) expressed in Escherichia coli using glutamine as substra...More data for this Ligand-Target Pair
TargetGlutaminase kidney isoform, mitochondrial(Homo sapiens (Human))
Calithera Biosciences Inc.
US Patent
Calithera Biosciences Inc.
US Patent
Affinity DataIC50: 1.40E+3nMAssay Description:No preinc (Column 4).More data for this Ligand-Target Pair