null
SMILES CN1CCN(CC1)c1nc(N)nc(n1)-c1ccncc1
InChI Key InChIKey=GBNBXYQUXOTKEI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 189355
Affinity DataKi: 3.19E+3nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
Affinity DataKi: 3.19E+3nM ΔG°: -6.97kcal/molepH: 7.4 T: 2°CAssay Description:Prior to the experiments, cell membranes were sedimented by a 10 min centrifugation at 4 °C
and 16 0009x g and resuspended in binding buffer (12...More data for this Ligand-Target Pair