null

SMILES CN1CCN(CC1)c1cc(ccn1)C(=O)Nc1cc2cc(ccc2cn1)-c1cnn(C)c1

InChI Key InChIKey=BQWWOBKMDWACGC-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 80 hits for monomerid = 293424   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1nMT: 2°CAssay Description:Briefly, recombinant DYRK1A kinase, ATP and Ser/Thr peptide 18 were prepared in 1× Kinase buffer to final concentrations of 0.19 μg/mL, 30 μ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.60nMT: 2°CAssay Description:Briefly, recombinant DYRK1A kinase, ATP and Ser/Thr peptide 18 were prepared in 1× Kinase buffer to final concentrations of 0.19 μg/mL, 30 μ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.5nMT: 2°CAssay Description:Briefly, recombinant DYRK1A kinase, ATP and Ser/Thr peptide 18 were prepared in 1× Kinase buffer to final concentrations of 0.19 μg/mL, 30 μ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.20nMT: 2°CAssay Description:Briefly, recombinant DYRK1A kinase, ATP and Ser/Thr peptide 18 were prepared in 1× Kinase buffer to final concentrations of 0.19 μg/mL, 30 μ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.40nMT: 2°CAssay Description:Briefly, recombinant DYRK1A kinase, ATP and Ser/Thr peptide 18 were prepared in 1× Kinase buffer to final concentrations of 0.19 μg/mL, 30 μ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.84E+3nMT: 2°CAssay Description:Briefly, recombinant GSK3β kinase, ATP and Ser/Thr peptide 09 are prepared in 1× Kinase buffer to final concentrations of 0.04 μg/mL, 46 &#...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  6.39E+3nMT: 2°CAssay Description:Briefly, recombinant GSK3β kinase, ATP and Ser/Thr peptide 09 are prepared in 1× Kinase buffer to final concentrations of 0.04 μg/mL, 46 &#...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  3.27E+3nMT: 2°CAssay Description:Briefly, recombinant GSK3β kinase, ATP and Ser/Thr peptide 09 are prepared in 1× Kinase buffer to final concentrations of 0.04 μg/mL, 46 &#...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.36E+3nMT: 2°CAssay Description:Briefly, recombinant GSK3β kinase, ATP and Ser/Thr peptide 09 are prepared in 1× Kinase buffer to final concentrations of 0.04 μg/mL, 46 &#...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  3.85E+3nMT: 2°CAssay Description:Briefly, recombinant GSK3β kinase, ATP and Ser/Thr peptide 09 are prepared in 1× Kinase buffer to final concentrations of 0.04 μg/mL, 46 &#...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN97Q3US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.84E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologiesa Div...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  6.39E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologiesa Div...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  3.27E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologiesa Div...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.36E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologiesa Div...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  3.85E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologiesa Div...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.40nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.60nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.5nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies-a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2862JRDUS Patent
TargetProto-oncogene Wnt-1(Homo sapiens (human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  46nMAssay Description:The screening assay for Wnt activity is described as follows. Reporter cell lines can be generated by stably transducing cancer cell lines (e.g., col...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetProto-oncogene Wnt-1(Homo sapiens (human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  55nMAssay Description:The screening assay for Wnt activity is described as follows. Reporter cell lines can be generated by stably transducing cancer cell lines (e.g., col...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetProto-oncogene Wnt-1(Homo sapiens (human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  45nMAssay Description:The screening assay for Wnt activity is described as follows. Reporter cell lines can be generated by stably transducing cancer cell lines (e.g., col...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetProto-oncogene Wnt-1(Homo sapiens (human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  51nMAssay Description:The screening assay for Wnt activity is described as follows. Reporter cell lines can be generated by stably transducing cancer cell lines (e.g., col...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetProto-oncogene Wnt-1(Homo sapiens (human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  55nMAssay Description:The screening assay for Wnt activity is described as follows. Reporter cell lines can be generated by stably transducing cancer cell lines (e.g., col...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.60nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.5nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.40nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.84E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Di...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  6.39E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Di...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  3.27E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Di...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.36E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Di...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  3.85E+3nMAssay Description:The GSK3β kinase assay is run using the Ser/Thr 09 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Di...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2H134DSUS Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.40nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8JR2US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8JR2US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.60nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8JR2US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.5nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8JR2US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.20nMAssay Description:The DYRKIA kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies—a Divis...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8JR2US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  6.39E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SJ1QR6
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  3.27E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SJ1QR6
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  1.36E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SJ1QR6
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Samumed, LLC

US Patent
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataEC50:  3.85E+3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SJ1QR6
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))TBA
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B06FXPubMed
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))TBA
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataIC50: 22nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B06FXPubMed
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))TBA
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6Q1VPubMed
TargetDual specificity protein kinase CLK2(Homo sapiens (Human))TBA
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6Q1VPubMed
TargetDual specificity protein kinase CLK3(Homo sapiens (Human))TBA
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
Affinity DataIC50: 20nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6Q1VPubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))TBA
LigandPNGBDBM293424(US10106527, Compound 10 | US10106527, Compound 142...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6Q1VPubMed
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