null
SMILES CC1Nc2cc(ccc2NC1=O)-c1cn(C)c(=O)c2[nH]ccc12
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 310876
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Genentech, Inc.; Constellation Pharmaceuticals Inc.
US Patent
Genentech, Inc.; Constellation Pharmaceuticals Inc.
US Patent
Affinity DataIC50: 110nMAssay Description:His/Flag epitope tagged BRD4 BD142-168 was cloned, expressed, and purified to. BRD4 binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair