null
SMILES Cn1cc(-c2ccc3NC(=O)CC(Nc3c2)c2cccs2)c2cc[nH]c2c1=O
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 310880
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Genentech, Inc.; Constellation Pharmaceuticals Inc.
US Patent
Genentech, Inc.; Constellation Pharmaceuticals Inc.
US Patent
Affinity DataIC50: 58nMAssay Description:His/Flag epitope tagged BRD4 BD142-168 was cloned, expressed, and purified to. BRD4 binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair