null

SMILES Cn1cc(-c2ccc(cc2)C(=O)N2CC(F)C2)c2cc[nH]c2c1=O

InChI Key InChIKey=LZEZGXBLBKUAKG-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 310884   

TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Genentech, Inc.; Constellation Pharmaceuticals Inc.

US Patent
LigandPNGBDBM310884(4-[4-(3-fluoroazetidine-1-carbonyl)phenyl]-6-methy...)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:His/Flag epitope tagged BRD4 BD142-168 was cloned, expressed, and purified to. BRD4 binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V98B5WUS Patent