null

SMILES Oc1ccc(cc1)C(=O)N[C@@H]1CNCCC[C@H]1OC(=O)c1cc(O)c(C2OC(=O)c3cccc(O)c23)c(O)c1

InChI Key InChIKey=RHPDVSROMSAMDQ-ZSUSVGCRSA-N

PDB links: 1 PDB ID contains inhibitors having a similarity of 90% to this monomer.

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Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 3226   

TargetProtein kinase C alpha type(Homo sapiens (Human))
Sphinx Laboratories

LigandPNGBDBM3226((3R,4R)-3-[(4-hydroxybenzene)amido]azepan-4-yl 3,5...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+4nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2M50PubMed
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
Sphinx Laboratories

LigandPNGBDBM3226((3R,4R)-3-[(4-hydroxybenzene)amido]azepan-4-yl 3,5...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:The activity of PKA, activated by cAMP, is measured by its ability to transfer phosphate from [gamma-32P]ATP to histone.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2M50PubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Sphinx Laboratories

LigandPNGBDBM3226((3R,4R)-3-[(4-hydroxybenzene)amido]azepan-4-yl 3,5...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+4nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2M50PubMed
TargetProtein kinase C beta type(Homo sapiens (Human))
Sphinx Laboratories

LigandPNGBDBM3226((3R,4R)-3-[(4-hydroxybenzene)amido]azepan-4-yl 3,5...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:PKC was assayed by quantitating the incorporation of 32P from [gamma-32P]ATP into histone type IIIs.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2M50PubMed