null
SMILES N#Cc1ccc2[nH]cc([C@@H]3CC[C@@H](CC3)N3CCc4ccccc4C3)c2c1
InChI Key InChIKey=LOEPSYRVNXADMM-TYKWCNGQSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50102010
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratories
Curated by ChEMBL
Wyeth-Ayerst Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:In vitro for its binding affinity for serotonin transporter RB5-HT-T in rat cortical membranesMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Affinity DataKi: 4.51nMAssay Description:Displacement of [3H]citalopram from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Affinity DataKi: 189nMAssay Description:Displacement of [3H]paroxetine from human SERT expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Wyeth-Ayerst Research Laboratories
Curated by ChEMBL
Wyeth-Ayerst Research Laboratories
Curated by ChEMBL
Affinity DataKi: 337nMAssay Description:Binding affinity at Alpha-1 adrenergic receptors on rat cortical membranes by [3H]prazosin displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Affinity DataKi: 424nMAssay Description:Displacement of [3H]WIN35428 from human DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in rat cortical membraneMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Institut für Interdisziplinäre Isotopenforschung
Curated by ChEMBL
Affinity DataKi: 1.43E+3nMAssay Description:Displacement of [3H]nisoxetine from human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair