null
SMILES CC(c1ccccc1)c1ccc(cc1)C(=O)NCc1c(C)cc(C)[nH]c1=O
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50110371
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.
Curated by ChEMBL
Constellation Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 795nMAssay Description:Inhibition of EZH2 Y641N mutant (unknown origin) using biotinylated nucleosome, H3K27me3 activator and [3H]-SAM incubated for 60 mins by top-count ba...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.
Curated by ChEMBL
Constellation Pharmaceuticals, Inc.
Curated by ChEMBL
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.
Curated by ChEMBL
Constellation Pharmaceuticals, Inc.
Curated by ChEMBL
TargetHistone-lysine N-methyltransferase EZH2(Homo sapiens (Human))
Constellation Pharmaceuticals, Inc.
Curated by ChEMBL
Constellation Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 153nMAssay Description:Inhibition of EZH2 (unknown origin) using biotinylated nucleosome, H3K27me3 activator and [3H]-SAM incubated for 60 mins by top-count based methodMore data for this Ligand-Target Pair