null
SMILES COc1ccc2nc(nc(NN3C(=O)C=C(C)C3=O)c2c1)-c1cccs1
InChI Key InChIKey=WAPBQFRODQBNJI-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50135483
TargetTranscription factor Jun(Homo sapiens (Human))
University of Texas Medical Branch
Curated by ChEMBL
University of Texas Medical Branch
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of AP-1-mediated transcriptional activation in human Jurkat cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 9.80E+3nMAssay Description:Induction of NFkappaB p65 nuclear translocation in HUVEC cells by immunostainingMore data for this Ligand-Target Pair
Affinity DataEC50: 4.20E+4nMAssay Description:Potentiation of TNFalpha-induced NFkappaB p65 nuclear translocation in HUVEC cells by immunostainingMore data for this Ligand-Target Pair