null
SMILES CCCOc1cccc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)c(C)n2)c1
InChI Key InChIKey=LSCCJMMALWILLE-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50150811
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center
Curated by ChEMBL
The University of Texas MD Anderson Cancer Center
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins...More data for this Ligand-Target Pair
TargetTranscription intermediary factor 1-alpha(Homo sapiens (Human))
The University of Texas MD Anderson Cancer Center
Curated by ChEMBL
The University of Texas MD Anderson Cancer Center
Curated by ChEMBL
Affinity DataEC50: 950nMAssay Description:Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ...More data for this Ligand-Target Pair