null
SMILES COCC1=C([C@@H](N(C(=O)NCCCN2CCC(CC2)c2cccc(NC(C)=O)c2)C(=O)N1)c1ccc(F)c(F)c1)C(=O)OC
InChI Key InChIKey=FWMHZWMPUWAUPL-NDEPHWFRSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50152456
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]SNAP 7941 from rat MCHR1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H]T226296 from rat recombinant MCH1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to rat MCH1 receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Lundbeck Research USA, Inc.
Curated by ChEMBL
Lundbeck Research USA, Inc.
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Displacement of [125I]HEAT from human recombinant adrenergic alpha1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+3nMAssay Description:Displacement of [3H]spiperone from human recombinant dopamine D2 receptorMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Abbott Laboratories
Curated by ChEMBL
Abbott Laboratories
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Concentration required to inhibit binding of [125I]-MCH radioligand to human Melanin-concentrating hormone receptor 1 in IMR-32 I3.4.2 cell membranesMore data for this Ligand-Target Pair