null
SMILES COc1cc(c(OC)cc1CN(C)C)-c1cc(C)c(=O)n(C)c1C
InChI Key InChIKey=ZEAWZAPWYCAHPL-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50183452
TargetBromodomain-containing protein 7(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Affinity DataIC50: 3.28E+3nMAssay Description:Inhibition of human N-terminal GST-tagged BRD7 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScreen ...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Affinity DataIC50: 5.96E+4nMAssay Description:Inhibition of human N-terminal GST-tagged BRD2-BD1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Affinity DataIC50: 134nMAssay Description:Inhibition of human N-terminal GST-tagged BRD9 isoform 1 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by Al...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Affinity DataIC50: 6.19E+4nMAssay Description:Inhibition of full-length MSR1 transfected in HEK293 cells by fluorimetryMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Boehringer Ingelheim RCV GmbH& Co KG
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human N-terminal GST-tagged BRD4-BD2 expressed in Escherichia coli using tetra-acetylated histone H4 measured after 60 mins by AlphaScr...More data for this Ligand-Target Pair