null
SMILES Cn1c(cc2sccc12)C(=O)Nc1ccccc1
InChI Key InChIKey=KIGYBJCTGONVIE-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50236398
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using biotinylated H3K4me1 peptide as substrate preincubated for 2...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
European Institute of Oncology IRCCS
Curated by ChEMBL
European Institute of Oncology IRCCS
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Homo sapiens (Human))
European Institute of Oncology
Curated by ChEMBL
European Institute of Oncology
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair