null
SMILES CC(C)CC(CC(C)C)C(=O)OCC1(CO)C\C(=C/c2cn(C)c3ccccc23)C(=O)O1
InChI Key InChIKey=ADNDQUKOVGKCGQ-UDWIEESQSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50244451
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]PDBu from RasGRP3 (unknown origin) expressed in cellsMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]PDBu from full length MBP-tagged human RasGRP3 expressed in Escherichia coli BL21 (DE3) after 5 mins by scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Displacement of [3H]PDBu from human recombinant PKCalpha expressed in Escherichia coli BL21-21-Gold (DE3)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Cancer Institute at Frederick
Curated by ChEMBL
National Cancer Institute at Frederick
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]PDBu from full length recombinant human PKCalpha expressed in baculovirus expression system after 5 mins by scintillation countin...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]PDBu from full length recombinant human PKCepsilon expressed in baculovirus expression system after 5 mins by scintillation count...More data for this Ligand-Target Pair