null
SMILES CN1CCc2c(C1)sc1nc([nH]c(=O)c21)-c1ccc(O)cc1
InChI Key InChIKey=IFZGKZCKUSRNJN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50251044
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center of Biotherapy
Curated by ChEMBL
Sichuan University and Collaborative Innovation Center of Biotherapy
Curated by ChEMBL
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of GST-tagged BRD4 bromodomain (unknown origin) using biotinylated histone H4KAc peptide (1 to 21 residues) as substrate by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center of Biotherapy
Curated by ChEMBL
Sichuan University and Collaborative Innovation Center of Biotherapy
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of His/thioredoxin-tagged human recombinant BRD4 bromodomain-1 (43 to 166 residues) expressed in Escherichia coli BL21 Star (DE3) pre-incu...More data for this Ligand-Target Pair