null
SMILES C(CN1CCOCC1)Cn1cc(-c2ccncc2)c2ccncc12
InChI Key InChIKey=MQUXYZGRXPUJHZ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50251476
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 109nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 7.58E+3nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
TargetNuclear factor of activated T-cells, cytoplasmic 1(Homo sapiens)
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataEC50: 6.96E+3nMAssay Description:Induction of nuclear translocation of human GFP-tagged NFATc1 expressed in virus infected primary human skeletal muscle myoblasts after 3 hrs by DAPI...More data for this Ligand-Target Pair