null
SMILES COc1cc(NC2CCN(C)CC2)c2cc(OC)c(OCCCN3CCCC3)cc2n1
InChI Key InChIKey=FJBOTWLVNUWQIU-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50281317
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias
Curated by ChEMBL
Universidad de Oviedo-Principado de Asturias
Curated by ChEMBL
Affinity DataIC50: 136nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias
Curated by ChEMBL
Universidad de Oviedo-Principado de Asturias
Curated by ChEMBL
Affinity DataIC50: 2.29E+3nMAssay Description:Inhibition of human DNMT1 using polydeoxyinosine polydeoxycytosine DNA as substrate after 15 mins in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair