null
SMILES COc1cc(cc(OC)c1C)[C@@H](O)[C@@H](CC1Cc2ccccc2C1)Cn1ccc(CCC(O)=O)c1
InChI Key InChIKey=USAXUWZJQPBEDO-ABYGYWHVSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50285779
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.190nMAssay Description:Antagonist activity at recombinant human LPA1 expressed in CHO cell membranes pretreated for 24 hrs prior to Fura-2-AM dye addition for 1 hr followed...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 2.30nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 0.5 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 0.740nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 0.740nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs at room temperature by scintillation counting methodMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 23nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs at 4 degC by scintillation counting methodMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 0.490nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 0.340nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs at 37 degC by scintillation counting methodMore data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Antagonist activity at recombinant human LPA1 expressed in CHO cell membranes pretreated for 24 hrs prior to Fura-2-AM dye addition for 1 hr followed...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 86nMAssay Description:Antagonist activity at recombinant human LPA1 expressed in CHO cells assessed as reduction in LPA-induced intracellular calcium level pretreated foll...More data for this Ligand-Target Pair
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
ONO Pharmaceutical Co., Ltd.
Curated by ChEMBL
Affinity DataKd: 1.30nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair